Flubromazolam is a triazole analog of flubromazepam and is a very high affinity, in-vitro benzodiazepine-related compound. It contains fluorine, bromine, and a methylated triazole substituent on its core benzodiazepine structure. Flubromazolam is a novel designer drug that is a synthetic version of the benzodiazepine class. Many designer drugs are former research drugs or drugs that were previously approved in other countries. Flubromazolam is a former research drug that did not make it to clinical trials. How strong is flubromazolam?
What is Flubromazolam?
Flubromazolam is a novel designer drug similar to flubromazolam that is described above. Like flubromazolam, flubromazolam is a triazole-benzodiazepine based derivative of benzodiazepine. Flubromazolam has been tested as a hypnotic drug. Its effects are similar to flubromazolam but flubromazolam has much more potent analgesic activity, so it is best used as an anesthetic rather than a sedative. Flubromazolam is considered a designer drug because it is produced using an improvised synthesis and has no existing medical uses. Flubromazolam is an analog of flubromazepam but has the fluorine, bromine and methylated triazole substituents replaced by a fluorine-fluorine moiety and a bromine-chloride moiety.
Flubromazolam has been on the market in Europe as a new class of benzodiazepines since 2008 but only recently became available in the United States in 2016. Despite this, Flubromazolam pallet is already one of the most toxic designer benzodiazepine derivatives. It is very potent, affecting a wide range of nervous system (neurological) systems that it can cause all in one pill. Flubromazolam is considered an extremely dangerous substance by the DEA. It has been labeled as an “abuse-deterrent” formulation in the form of fluconazole citrate, but this was later rescinded due to the fact that such claims were never made by the manufacturer. Flubromazolam is also considered a Schedule IV drug by the DEA. It is classified as a Category C drug for both in vitro and in vivo toxicity.Buy benzodiazepines online
Flubromazolam’s mechanisms of action involve binding to the benzodiazepine site of the GABA receptor. It is believed to have the same effects of a benzodiazepine or a mixed benzodiazepine and phenazine with the central nervous system relaxant effects. Flubromazolam acts in many ways on the brain such as atropine, N-methyl-D-aspartate receptor agonism, and NMDA receptor antagonism. Many of the GABA receptors are important in the nervous system such as the NMDA receptors. NMDAR is known for its control of glutamate, which is a neurotransmitter essential in brain function. How strong is flubromazolam which has a very high-affinity binding to NMDA receptors? It also binds to the serotonin 5-HT2a and 5-HT1a receptors, where it has a psychostimulant effect.- Deadly Designer Benzodiazepine
Flubromazolam’s potency and euphoric effects may provide a pleasurable experience at higher doses, but the resulting drowsiness and potential respiratory depression can lead to an overdose death. Flubromazolam affects the same brain receptors as other benzodiazepine derivatives such as flubromazolaml, methoxydiazepam, and methediazepam. Flubromazolam can block the receptor-mediated effects of flubromazolaml, so users may believe that they are getting a full-spectrum sedative effect. However, flubromazolam may have similar or even worse effects when it is taken in conjunction with other drugs such as alcohol, cocaine, or methoxydiazepam.
Flubromazolam’s Effects on the Brain
Flubromazolam is an orally active benzodiazepine compound. It has benzodiazepine-type effects similar to a class of potent benzodiazepine’s including alprazolam, alprazolamlopride, and temazepam. In humans, flubromazolam has been shown to cause profound sedation with the rapid onset of sedation causing drowsiness and muscle relaxation. These effects can last up to four hours after the pill is ingested. These drowsiness and muscle relaxation effects can persist for a period of time and can be severe enough to induce a high level of anxiety. While the body’s natural relaxation response may aid some people to get off the drug, it may cause a person to become angry and agitated. The peak blood pressure is 250/160 mmHg and the peak heart rate is 105 bpm.
Flubromazolam’s Effects on the Body
Flubromazolam has a very potent binding affinity for the benzodiazepine site of the GABA receptors. At low doses, flubromazolam pellets can produce symptoms similar to those of benzodiazepines such as euphoria, anxiety, sedation, and dizziness. At high doses, however, flubromazolam has much more potent effects. Flubromazolam produces effects similar to all benzodiazepines. It produces dissociative effects which are much stronger than those of benzodiazepines. In addition, it produces anxiolytic, anticonvulsant, hypnotic, antimuscarinic, antidiarrheal, sedative, analgesic, and dissociative effects at very high doses. Flubromazolam is a very potent dissociative, antimuscarinic, and anxiolytic drug.
How strong is flubromazolam, Flubromazolam is an extremely dangerous and lethal designer benzodiazepine derivative. Users who are abusing Flubromazolam should know that they are taking a very dangerous drug.